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1

La communication sociétale des entreprises de travail temporaire face au stress des intérimaires lié à la précarité du secteur d’activité

Robaa, Guillaume

Journal:

RIMHE : Revue Interdisciplinaire Management, Homme(s) & Entreprise

Year:

2018

Language:

french

File:

PDF, 823 KB

french, 2018

2

Characterization of histone deacetylase 8 (HDAC8) selective inhibition reveals specific active site structural and functional determinants

Marek, Martin, Shaik, Tajith Baba, Heimburg, Tino, Chakrabarti, Alokta, LANCELOT, Julien, Ramos Morales, Elizabeth, Da Veiga, Cyrielle, Kalinin, Dmitrii V., Melesina, Jelena, Robaa, Dina, Schmidtkunz,

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 2.07 MB

english, 2018

3

A Novel Non-phenolic Dibenzazecine Derivative with Nanomolar Affinities for Dopamine Receptors

Dina Robaa, Shams ElDin AbulAzm, Jochen Lehmann, Christoph Enzensperger

Journal:

Chemistry & Biodiversity

Year:

2011

Language:

english

File:

PDF, 179 KB

english, 2011

4

Enantiomerically Pure 2-Methyltetrahydro-3-benzazepin-1-ols Selectively Blocking GluN2B Subunit Containing N -Methyl- d -aspartate Receptors

Tewes, Bastian, Frehland, Bastian, Schepmann, Dirk, Robaa, Dina, Uengwetwanit, Tanaporn, Gaube, Friedemann, Winckler, Thomas, Sippl, Wolfgang, Wünsch, Bernhard

Journal:

Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 4.43 MB

english, 2015

5

Chemically Induced Degradation of Sirtuin 2 (Sirt2) by a Proteolysis Targeting Chimera (PROTAC) Based on Sirtuin Rearranging Ligands (SirReals)

Schiedel, Matthias, Herp, Daniel, Hammelmann, Sören, Swyter, Sören, Lehotzky, Attila, Robaa, Dina, Oláh, Judit, Ovádi, Judit, Sippl, Wolfgang, Jung, Manfred

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.05 MB

english, 2017

6

Proteolysis targeting chimeras (PROTACs) for epigenetics research

Vogelmann, Anja, Robaa, Dina, Sippl, Wolfgang, Jung, Manfred

Journal:

Current Opinion in Chemical Biology

Year:

2020

File:

PDF, 1.30 MB

2020

7

Residues at the Indole-NH of LE300 Modulate Affinities and Selectivities for Dopamine Receptors

Dina Robaa, Robert Kretschmer, Oliver Siol, Shams ElDin AbulAzm, ElSayeda ElKhawass, Jochen Lehmann, Christoph Enzensperger

Journal:

Archiv der Pharmazie

Year:

2011

Language:

english

File:

PDF, 289 KB

english, 2011

8

A study of solar radiation climate at Cairo urban area, Egypt and its environs

Journal:

International Journal of Climatology

Year:

2006

Language:

english

File:

PDF, 395 KB

english, 2006

9

Human climates of Egypt

S. M. Robaa, H. M. Hasanean

Journal:

International Journal of Climatology

Year:

2007

Language:

english

File:

PDF, 1.84 MB

english, 2007

10

A study of ultraviolet solar radiation at Cairo urban area, Egypt

Journal:

Year:

2004

Language:

english

File:

PDF, 347 KB

english, 2004

11

Evaluation of sunshine duration from cloud data in Egypt

Journal:

Year:

2008

Language:

english

File:

PDF, 563 KB

english, 2008

12

Validation of the existing models for estimating global solar radiation over Egypt

Journal:

Energy Conversion and Management

Year:

2009

Language:

english

File:

PDF, 218 KB

english, 2009

13

Urban–rural solar radiation loss in the atmosphere of Greater Cairo region, Egypt

Journal:

Energy Conversion and Management

Year:

2009

Language:

english

File:

PDF, 607 KB

english, 2009

14

Dopamine Receptor Ligands. Part 18:(1) Modification of the Structural Skeleton of Indolobenzazecine-Type Dopamine Receptor Antagonists

Robaa, Dina, Enzensperger, Christoph, Abul Azm, Shams El Din, El Khawass, El Sayeda, El Sayed, Ola, Lehmann, Jochen

Journal:

Journal of Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 783 KB

english, 2010

15

Chiral Indolo[3,2- f ][3]benzazecine-Type Dopamine Receptor Antagonists: Synthesis and Activity of Racemic and Enantiopure Derivatives

Robaa, Dina, Enzensperger, Christoph, ElDin AbulAzm, Shams, Hefnawy, Mohamed M., El-Subbagh, Hussein I., Wani, Tanveer A., Lehmann, Jochen

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 926 KB

english, 2011

16

A study of ultraviolet solar radiation at Cairo urban area, Egypt

Journal:

Year:

2004

Language:

english

File:

PDF, 347 KB

english, 2004

17

Mind the Methyl: Methyllysine Binding Proteins in Epigenetic Regulation

Wagner, Tobias, Robaa, Dina, Sippl, Wolfgang, Jung, Manfred

Journal:

Year:

2014

Language:

english

File:

PDF, 4.80 MB

english, 2014

18

Pyrido- and benzisothiazolones as inhibitors of histone acetyltransferases (HATs)

Furdas, S. D., Hoffmann, I., Robaa, D., Herquel, B., Malinka, W., Świątek, P., Akhtar, A., Sippl, W., Jung, M.

Journal:

Year:

2014

Language:

english

File:

PDF, 297 KB

english, 2014

19

Peptide Backbone Conformation Affects the Substrate Preference of Protein Arginine Methyltransferase I

Kölbel, Knut, Ihling, Christian, Kühn, Uwe, Neundorf, Ines, Otto, Silke, Stichel, Jan, Robaa, Dina, Beck-Sickinger, Annette G., Sinz, Andrea, Wahle, Elmar

Journal:

Year:

2012

Language:

english

File:

PDF, 1.29 MB

english, 2012

20

Analysis of the Resistance of Hepatitis C Virus NS5B Polymerase Inhibitors via Docking and Molecular Dynamics Simulation

Uengwetwanit, Tanaporn, Robaa, Dina, Sippl, Wolfgang

Journal:

Molecular Informatics

Year:

2015

Language:

english

File:

PDF, 1.73 MB

english, 2015

21

Evaluation of Homobivalent Carbolines as Designed Multiple Ligands for the Treatment of Neurodegenerative Disorders

Otto, Robert, Penzis, Robert, Gaube, Friedemann, Adolph, Oliver, Föhr, Karl J., Warncke, Paul, Robaa, Dina, Appenroth, Dorothea, Fleck, Christian, Enzensperger, Christoph, Lehmann, Jochen, Winckler, T

Journal:

Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 434 KB

english, 2015

22

Molecular Combination of the Dopamine and Serotonin Scaffolds Yield in Novel Antipsychotic Drug Candidates - Characterization by in vivo Experiments

Schulze, M., Siol, O., Robaa, D., Mueller, F.K., Enzensperger, C., Fleck, C., Lehmann, J.

Journal:

Arzneimittelforschung

Year:

2012

Language:

english

File:

PDF, 374 KB

english, 2012

23

Homology Modeling of Parasite Histone Deacetylases to Guide the Structure-Based Design of Selective Inhibitors

Melesina, Jelena, Robaa, Dina, Pierce, Raymond J., Romier, Christophe, Sippl, Wolfgang

Journal:

Journal of Molecular Graphics and Modelling

Year:

2015

Language:

english

File:

PDF, 2.24 MB

english, 2015

24

Benzo[7]annulene-based GluN2B selective NMDA receptor antagonists: Surprising effect of a nitro group in 2-position

Gawaskar, Sandeep, Schepmann, Dirk, Bonifazi, Alessandro, Robaa, Dina, Sippl, Wolfgang, Wünsch, Bernhard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 744 KB

english, 2015

25

KATching-Up on Small Molecule Modulators of Lysine Acetyltransferases

Simon, Roman P., Robaa, Dina, Alhalabi, Zayan, Sippl, Wolfgang, Jung, Manfred

Journal:

Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.73 MB

english, 2016

26

Substituted 2-(2-aminopyrimidin-4-yl)pyridine-4-carboxylates as potent inhibitors of JumonjiC domain-containing histone demethylases

Roatsch, Martin, Robaa, Dina, Pippel, Martin, Nettleship, Joanne E, Reddivari, Yamini, Bird, Louise E, Hoffmann, Inga, Franz, Henriette, Owens, Raymond J, Schüle, Roland, Flaig, Ralf, Sippl, Wolfgang,

Journal:

Future Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.31 MB

english, 2016

27

Structure-Based Design and Synthesis of Novel Inhibitors Targeting HDAC8 from Schistosoma mansoni for the Treatment of Schistosomiasis

Heimburg, Tino, Chakrabarti, Alokta, Lancelot, Julien, Marek, Martin, Melesina, Jelena, Hauser, Alexander-Thomas, Shaik, Tajith B., Duclaud, Sylvie, Robaa, Dina, Erdmann, Frank, Schmidt, Matthias, Rom

Journal:

Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 6.81 MB

english, 2016

28

Stereospecific capillary electrophoresis assays using pentapeptide substrates for the study of aspergillus nidulans methionine sulfoxide reductase a and mutant enzymes

Zhu, Qingfu, El-Mergawy, Rabab G., Zhou, Yuzhen, Chen, Chunyang, Heinemann, Stefan H., Schönherr, Roland, Robaa, Dina, Sippl, Wolfgang, Scriba, Gerhard K. E.

Journal:

ELECTROPHORESIS

Year:

2016

Language:

english

File:

PDF, 1011 KB

english, 2016

29

Some aspects of the urban climates of Greater Cairo Region, Egypt

Journal:

International Journal of Climatology

Year:

2013

Language:

english

File:

PDF, 308 KB

english, 2013

30

Identification and Structure-Activity Relationship Studies of Small-Molecule Inhibitors of the Methyllysine Reader Protein Spindlin1

Robaa, Dina, Wagner, Tobias, Luise, Chiara, Carlino, Luca, McMillan, Joel, Flaig, Ralf, Schüle, Roland, Jung, Manfred, Sippl, Wolfgang

Journal:

Year:

2016

Language:

english

File:

PDF, 1.47 MB

english, 2016

31

Synthesis, biological characterisation and structure activity relationships of aromatic bisamidines active against Plasmodium falciparum

Sauer, B., Skinner-Adams, T.S., Bouchut, A., Chua, M.J., Pierrot, C., Erdmann, F., Robaa, D., Schmidt, M., Khalife, J., Andrews, K.T., Sippl, W.

Journal:

European Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.27 MB

english, 2017

32

The Current State of NAD + -Dependent Histone Deacetylases (Sirtuins) as Novel Therapeutic Targets

Schiedel, Matthias, Robaa, Dina, Rumpf, Tobias, Sippl, Wolfgang, Jung, Manfred

Journal:

Medicinal Research Reviews

Year:

2017

Language:

english

File:

PDF, 1.28 MB

english, 2017

33

Lysine Deacetylase Inhibitors in Parasites: Past, Present, and Future Perspectives

Hailu, Gebremedhin S., Robaa, Dina, Forgione, Mariantonietta, Sippl, Wolfgang, Rotili, Dante, Mai, Antonello

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.12 MB

english, 2017

34

Evolutionary relationships among protein lysine deacetylases of parasites causing neglected diseases

Scholte, Larissa L.S., Mourão, Marina M., Pais, Fabiano Sviatopolk-Mirsky, Melesina, Jelena, Robaa, Dina, Volpini, Angela C., Sippl, Wolfgang, Pierce, Raymond J., Oliveira, Guilherme, Nahum, Laila A.

Journal:

Infection, Genetics and Evolution

Year:

2017

Language:

english

File:

PDF, 1.06 MB

english, 2017

35

Photochromic histone deacetylase inhibitors based on dithienylethenes and fulgimides

Wutz, Daniel-Fabian, Gluhacevic, Dino, Chakrabarti, Alokta, karin.schmidtkunz, Karin, Robaa, Dina, Erdmann, Frank, Romier, Christophe, Sippl, Wolfgang, Jung, Manfred, Koenig, Burkhard

Journal:

Organic & Biomolecular Chemistry

Year:

2017

Language:

english

File:

PDF, 1.12 MB

english, 2017

36

Design, Synthesis, Pharmacological Evaluation and Docking Studies of GluN2B-Selective NMDA Receptor Antagonists with a Benzo[7]annulen-7-amine Scaffold

Gawaskar, Sandeep, Temme, Louisa, Schreiber, Julian A., Schepmann, Dirk, Bonifazi, Alessandro, Robaa, Dina, Sippl, Wolfgang, Strutz-Seebohm, Nathalie, Seebohm, Guiscard, Wünsch, Bernhard

Journal:

Year:

2017

Language:

english

File:

PDF, 1.10 MB

english, 2017

37

Evaluation of human-induced vibration of continuous footbridges

El-Robaa, Ahmed, Gaawan, Sameh, Malek, Charles, Feltrin, G.

Journal:

MATEC Web of Conferences

Year:

2015

Language:

english

File:

PDF, 418 KB

english, 2015

38

Structure-based design and biological characterization of selective histone deacetylase 8 (HDAC8) inhibitors with anti-neuroblastoma activity

Heimburg, Tino, Kolbinger, Fiona R., Zeyen, Patrik, Ghazy, Ehab, Herp, Daniel, Schmidtkunz, Karin, Melesina, Jelena, Shaik, Tajith Baba, Erdmann, Frank, Schmidt, Matthias, Romier, Christophe, Robaa, D

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.86 MB

english, 2017

39

Structure-activity studies on N -Substituted tranylcypromine derivatives lead to selective inhibitors of lysine specific demethylase 1 (LSD1) and potent inducers of leukemic cell differentiation

Schulz-Fincke, Johannes, Hau, Mirjam, Barth, Jessica, Robaa, Dina, Willmann, Dominica, Kürner, Andreas, Haas, Julian, Greve, Gabriele, Haydn, Tinka, Fulda, Simone, Lübbert, Michael, Lüdeke, Steffen, B

Journal:

European Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.96 MB

english, 2017

40

Hydroxymethyl bioisosteres of phenolic GluN2B-selective NMDA receptor antagonists: Design, synthesis and pharmacological evaluation

Temme, Louisa, Frehland, Bastian, Schepmann, Dirk, Robaa, Dina, Sippl, Wolfgang, Wünsch, Bernhard

Journal:

European Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.49 MB

english, 2017

41

Epigenetic small molecule modulators of histone and DNA methylation

Hauser, Alexander-Thomas, Robaa, Dina, Jung, Manfred

Journal:

Current Opinion in Chemical Biology

Year:

2018

Language:

english

File:

PDF, 908 KB

english, 2018

42

Activity of bromodomain protein inhibitors/binders against asexual-stage Plasmodium falciparum parasites

Chua, Ming Jang, Robaa, Dina, Skinner-Adams, Tina S., Sippl, Wolfgang, Andrews, Katherine T.

Journal:

International Journal for Parasitology Drugs and Drug Resistance

Year:

2018

Language:

english

File:

PDF, 528 KB

english, 2018

43

Synthesis, crystallization studies and in vitro characterization of novel cinnamic acid derivatives as SmHDAC8 inhibitors for the treatment of Schistosomiasis

Bayer, Theresa, Chakrabarti, Alokta, Lancelot, Julien, Shaik, Tajith B., Hausmann, Kristin, Melesina, Jelena, Schmidtkunz, Karin, Marek, Martin, Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Romier,

Journal:

Year:

2018

Language:

english

File:

PDF, 1.64 MB

english, 2018

44

Opening the Selectivity Pocket in the Human Lysine Deacetylase Sirtuin2 - New Opportunities, New Questions

Robaa, Dina, Monaldi, Daria, Wössner, Nathalie, Norio,, Kudo,, Rumpf, Tobias, Schiedel, Matthias, Yoshida, Minoru, Jung, Manfred

Journal:

The Chemical Record

Year:

2018

Language:

english

File:

PDF, 2.63 MB

english, 2018

45

Design of selective histone deacetylase inhibitors: rethinking classical pharmacophore

Melesina, Jelena, Praetorius, Lucas, Simoben, Conrad V, Robaa, Dina, Sippl, Wolfgang

Journal:

Future Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 168 KB

english, 2018

46

Muscle Carnitine Palmitoyltransferase II Deficiency: A Review of Enzymatic Controversy and Clinical Features

Lehmann, Diana, Motlagh, Leila, Robaa, Dina, Zierz, Stephan

Journal:

International Journal of Molecular Sciences

Year:

2017

Language:

english

File:

PDF, 1.10 MB

english, 2017

47

A Novel Class of Schistosoma mansoni Histone Deacetylase 8 (HDAC8) Inhibitors Identified by Structure-Based Virtual Screening and In Vitro Testing

Simoben, Conrad, Robaa, Dina, Chakrabarti, Alokta, Schmidtkunz, Karin, Marek, Martin, Lancelot, Julien, Kannan, Srinivasaraghavan, Melesina, Jelena, Shaik, Tajith, Pierce, Raymond, Romier, Christophe,

Journal:

Year:

2018

Language:

english

File:

PDF, 4.34 MB

english, 2018

48

Pharmacogenetic Aspects of the Interaction of AT1 Receptor Antagonists With ATP-Binding Cassette Transporter ABCG2

Ripperger, Anne, Krischer, Anna, Robaa, Dina, Sippl, Wolfgang, Benndorf, Ralf A.

Journal:

Frontiers in Pharmacology

Year:

2018

Language:

english

File:

PDF, 3.77 MB

english, 2018

49

The influence of two land-surface hydrology schemes on the regional climate of Africa using the RegCM4 model

Anwar, Samy A., Zakey, A.S., Robaa, S.M., Abdel Wahab, M. M.

Journal:

Theoretical and Applied Climatology

Year:

2018

Language:

english

File:

PDF, 9.45 MB

english, 2018

50

Front Cover: Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as Sm HDAC8 Inhibitors for the Treatment of Schistosomiasis (ChemMedChem 15/2018)

Bayer, Theresa, Chakrabarti, Alokta, Lancelot, Julien, Shaik, Tajith B., Hausmann, Kristin, Melesina, Jelena, Schmidtkunz, Karin, Marek, Martin, Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Romier,

Journal:

Year:

2018

File:

PDF, 498 KB

2018